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프로그램 비교

검색으로 10,000+ 프로그램 중 최대 5개를 골라 PK/PD · 독성 · 임상을 나란히 비교합니다. · 다음 갱신 D-13 · 마지막 7월 13일

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항목
ADCPhase 2
Selumetinib (Selumetinib)
AstraZeneca·Non-Small Cell Lung Cancer
ORR 19.7%
Overview
Program
Selumetinib
Overview
Company
AstraZeneca
Overview
Modality
ADC
Overview
Target
Non-Small Cell Lung Cancer
Overview
Indication
Advanced Pancreatic Ductal Adenocarcinoma; Metastatic Pancreatic Ductal Adenocarcinoma
Overview
Phase
PHASE_2
Overview
Status
RECRUITING
MoA
Mechanism
target poor prognosis KMT2A-rearranged RAS pathway
MoA
Biomarker
EGFR)-mutated advanced non-small cell lung cancer (NSCLC) follow
PK/PD
Species
Mouse, Human
PK/PD
Animal (cat.)
Human, Mouse, In vitro
PK/PD
Experiment
PK
Toxicology
Species
Mouse, Human
Toxicology
Animal (cat.)
Human, Mouse, In vitro
Toxicology
Major finding
Osimertinib plus selumetinib in patients with EGFR-mutated advanced NSCLC with BRAF alterations post-progression on first-line osimertinib: ORCHARD.. ORCHARD (NCT03944772) was a phase II, biomarker-matched, platform study designed to characterise resistance mechanisms and evaluate novel drug combinations in patients with epidermal growth factor receptor (EGFR)-mutated advanced non-small cell lung …
Clinical
Primary efficacy
ORR 19.7%
Clinical
ORR
19.7%
Clinical
Result source
ClinicalTrials.gov NCT04924608
Clinical
Data Tier / Score
A · 41
Clinical
Program phase
PHASE_2
Clinical
Clinical sync
2026년 7월 9일 (5일 전)