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프로그램 비교

검색으로 10,000+ 프로그램 중 최대 5개를 골라 PK/PD · 독성 · 임상을 나란히 비교합니다. · 다음 갱신 D-13 · 마지막 7월 13일

현재 선택: 2 · Data Tier에서 열림

프로그램 상세에서 관심 등록 후 2개 이상 모으면 여기서 한 번에 비교할 수 있습니다.

API CSV22행 · 2개 프로그램

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항목
AntibodyFDAApproved
daratumumab (Darzalex)
Janssen·CD38
ORR 80%·t½ 0.5 h
AntibodyApproved
Carfilzomib (Carfilzomib)
Pfizer·Multiple Myeloma
ORR 97%·t½ 1 h
Overview
Program
Darzalex (daratumumab)Carfilzomib
Overview
Company
JanssenPfizer
Overview
Modality
ANTIBODYANTIBODY
Overview
Target
CD38Multiple Myeloma
Overview
Indication
Multiple myelomaMultiple Myeloma
Overview
Phase
APPROVEDAPPROVED
Overview
Status
APPROVEDRECRUITING
MoA
Mechanism
CD38 targeting, Fc effector function, immunomodulationtargets, we performed gene set enrichment analysis on three publicly available HB datasets and found consistent activation of the proteasome pathway
MoA
Biomarker
CD38 expression on plasma cellsbiomarker and therapeutic target
PK/PD
Half-life
0.5 h1 h
PK/PD
Species
MouseMouse
PK/PD
Animal (cat.)
MouseMouse, In vitro
PK/PD
Experiment
pharmacokineticPD
Toxicology
Species
MouseMouse, Rat, Rabbit
Toxicology
Animal (cat.)
UnknownMouse, Rat, Monkey
Toxicology
Major finding
Hepatotoxicity Hepatotoxicity includes alanine aminotransferase increased, aspartate aminotinterstitial lung disease, occurred in approximately 2% of patients who received Kyprolis
Clinical
Primary efficacy
ORR 80%ORR 97%
Clinical
ORR
>80% in combo regimens97.0%
Clinical
Result source
POLLUX/CASTORClinicalTrials.gov NCT03412565
Clinical
Data Tier / Score
S · 94C · 70
Clinical
Program phase
APPROVEDAPPROVED
Clinical
Clinical sync
2026년 7월 8일 (6일 전)2026년 7월 4일 (9일 전)