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프로그램 비교

검색으로 10,000+ 프로그램 중 최대 5개를 골라 PK/PD · 독성 · 임상을 나란히 비교합니다. · 다음 갱신 D-13 · 마지막 7월 13일

현재 선택: 4

프로그램 상세에서 관심 등록 후 2개 이상 모으면 여기서 한 번에 비교할 수 있습니다.

API CSV25행 · 4개 프로그램

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항목
ADCFDAApproved
disitamab vedotin (Disitamab Vedotin, RC48)
RemeGen·HER2
ORR 50%·t½ ~5 days
ADCFDAApproved
enfortumab vedotin (Padcev)
Astellas / Seagen·Renal Pelvis and Ureter Urothelial…
ORR 44%·t½ 3.6 h
CGTFDAApproved
nadofaragene firadenovec (Adstiladrin, rAd-IFNα/Syn3, nadofaragene firadenovec-vncg)
Ferring Pharmaceuticals·IFNα2b (adenoviral)
ORR 55%
AntibodyPhase 3
Fluorouracil (Fluorouracil)
Janssen Research & Development, LL…·Muscle Invasive Bladder Carcinoma
ORR 80%
Overview
Program
Disitamab Vedotin (RC48)Enfortumab VedotinAdstiladrin (nadofaragene firadenovec)Fluorouracil
Overview
Company
RemeGenAstellas / SeagenFerring PharmaceuticalsJanssen Research & Development, LLC
Overview
Modality
ADCADCCGTANTIBODY
Overview
Target
HER2Renal Pelvis and Ureter Urothelial CarciIFNα2b (adenoviral)Muscle Invasive Bladder Carcinoma
Overview
Indication
HER2+ urothelial, gastric, breastMetastatic Bladder Urothelial Carcinoma; Metastatic Renal Pelvis and Ureter Urothelial CarcinomaHigh-risk BCG-unresponsive non-muscle invasive bladder cancer (NMIBC)Advanced or Metastatic Colorectal Cancer
Overview
Phase
APPROVEDAPPROVEDAPPROVEDPHASE_3
Overview
Status
ACTIVERECRUITINGAPPROVEDRECRUITING
MoA
Mechanism
HER2-mediated delivery of MMAEADC, while the AKR1C1-WWP2 axis promotes extracellular vesicle-mediated ADC export and clearance, thereby reducing intracellular payload accumulationAdenoviral transduction of urothelium → local IFNα2b expression → antitumor immunityinhibits GC cell proliferation and induces apoptosis by regulating cell-cycle checkpoints and inhibiting oncogenic pathway
MoA
Biomarker
HER2 expressionbiomarkers are limitedCR rate, duration of responsebiomarker for metabolic state, B-cell/TLS-associated immune features, and vulnerability to DNA damage-based t
PK/PD
Half-life
~5 days3.6 h
PK/PD
Species
MouseMouse, HumanMouseMouse
PK/PD
Animal (cat.)
Mouse, In vitroHuman, Mouse, In vitroMouse, In vitroMouse
PK/PD
Experiment
PDPharmacokineticpharmacodynamicPD
Toxicology
Species
MouseCynomolgus monkey, Mouse, Rat, HumanCynomolgus monkey, MouseMouse, Human
Toxicology
Animal (cat.)
Mouse, In vitroMouse, Rat, NHPNHPHuman
Toxicology
Major finding
thrombocytopenia, demonstrated for Kadcyla and EnhertuInterstitial Lung Disease (ILD): Severe, life-threatening or fatal pneumonitis/ILD may occurthrombocytopenia, inflammation of the esophagus, stomach, and small bowel
Clinical
Primary efficacy
ORR 50%ORR 44%ORR 55%ORR 80%
Clinical
ORR
~50% in HER2+ UC39%55%80.0%
Clinical
PFS
6.9 mo5.8
Clinical
OS
12.4100
Clinical
Result source
RC48-C009ClinicalTrials.gov NCT03219333ClinicalTrials.gov NCT02773849ClinicalTrials.gov NCT04430738
Clinical
Data Tier / Score
S · 89B · 88C · 78C · 70
Clinical
Program phase
APPROVEDAPPROVEDAPPROVEDPHASE_3
Clinical
Dose / schedule
q2wq3 months (label)
Clinical
Clinical sync
2026년 7월 8일 (6일 전)2026년 7월 4일 (9일 전)2026년 7월 12일 (1일 전)2026년 7월 4일 (9일 전)